Etomidate

  • Mechanism of Action: Facilitates inhibitory neurotransmission by enhancing the function (GABAA) receptors.
  • Pharmacokinetics: Effects of a single bolus dose are terminated by redistribution.
  • Primary Uses: Induction of anesthesia in patients with cardiovascular problems.
  • Advantages: Short acting and potent, with CVS and RS stability, suitable for elderly and shocked patients.
  • Adverse Effects:
    • Cause nausea and vomiting.
    • Adrenal suppression.
    • A single dose suppresses adrenal steroid synthesis.
    • No analgesic properties.