Ketamine

  • Mechanism of Action: Mainly attributed to noncompetitive antagonism of NMDA receptors in the CNS.
  • Pharmacokinetics: Unconsciousness in 30 to 60 s after an IV. Terminated by redistribution in 15 to 20 minutes.
  • Primary Uses: Induction of general anesthesia. Analgesia.
  • Advantages:
    • CVS stability makes it suitable for shocked patients.
    • Preservation of airway reflexes & less respiratory depression.
    • Potent bronchodilator.
  • Adverse Effects:
    • ↑ HR, and BP not good for hypertensive patient.
    • ↑ salivation, PONV, agitation & hallucinations.
    • Contraindicated in patients with head trauma.